Product Name: BX-912
Subtitle: PDK1 inhibitor,potent and ATP-competitive
Biological Activity: Biological Activity of BX-912Description BX-912 is a potent, ATP-competitive inhibitor of PDK-1 with IC50 value of 26 nM. Targets PDK-1 IC50 26 nM
SMLES: C1CCN(C1)C(=O)NC2=CC=CC(=C2)NC3=NC=C(C(=N3)NCCC4=CN=CN4)Br
CAS NO: 1408064-71-0
Standard In CHIKey: Antibody-drug Conjugate_ADC Related inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C20H23BrN8O
M.Wt: 471.35
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/257/1/439
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO > 10 mM
Storage:
Purity: >98%
Chemical Name: N-[3-[[5-bromo-4-[2-(1H-imidazol-5-yl)ethylamino]pyrimidin-2-yl]amino]phenyl]pyrrolidine-1-carboxamide

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