Product Name: IRL-2500
Subtitle:
Biological Activity: Biological Activity of IRL-2500Potent endothelin receptor antagonist; shows some selectivity for ETB receptors (IC50 values are 1.3 and 94 nM for ETB and ETA receptors respectively). Inhibits ETB receptor-mediated blood pressure increase and renal vascula
SMLES: O=C([C@@H](CC1=CC=C(C2=CC=CC=C2)C=C1)N(C)C(C3=CC(C)=CC(C)=C3)=O)N[C@H](C(O)=O)CC4=CNC5=CC=CC=C45
CAS NO: 1675201-83-8
Standard In CHIKey: Fatty Acid Synthase FAS) inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C36H35N3O4
M.Wt: 573.69
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/265/2/1001
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in 1eq. NaOH
Storage: Desiccate at RT
Purity: >98%
Chemical Name: N-3-[1,1-Biphenyl]-4-yl-N-(3,5-dimethylbenzoyl)-N-methyl-D-alanyl-L-tryptophan