Product Name: Linagliptin (BI-1356)
Subtitle: DDP-4 inhibitor,highly potent and competitive
Biological Activity: Biological Activity of Linagliptin (BI-1356)Description Linagliptin is a highly potent, competitive inhibitor of dipeptidyl-peptidase 4 (DDP-4) with IC50 value of 1 nM. Targets DDP-4 IC50 1 nM
SMLES: CC#CCN1C2=C(N=C1N3CCCC(C3)N)N(C(=O)N(C2=O)CC4=NC5=CC=CC=C5C(=N4)C)C
CAS NO: 1032568-63-0
Standard In CHIKey: c-Myc inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C25H28N8O2
M.Wt: 472.5
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/258/1/74
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO > 10 mM
Storage:
Purity: >98%
Chemical Name: 8-[(3R)-3-aminopiperidin-1-yl]-7-but-2-ynyl-3-methyl-1-[(4-methylquinazolin-2-yl)methyl]purine-2,6-dione