Product Name: MK-2894
Subtitle: EP4 receptor inhibitor
Biological Activity: Biological Activity of MK-2894Description MK-2894 is a highly potent and selective inhibitor of EP4 receptor with IC50 value of 2.5 nM. Targets EP4 receptor IC50 2.5 nM (Ki=0.56±0.1 nM）
SMLES: Cc1c(c(c(s1)C)C(=O)NC2(CC2)c3ccc(cc3)C(=O)O)Cc4ccc(cc4)C(F)(F)F
CAS NO: 266359-93-7
Standard In CHIKey: Phospholipase inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C25H22F3NO3S
M.Wt: 473.51
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/254/1/98
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO
Storage:
Purity: >98%
Chemical Name: 4-{1-[({2,5-Dimethyl-4-[4-(trifluoromethyl)benzyl]-3-thienyl}carbonyl)amino]cyclopropyl}benzoic acid