Product Name: PIK-75
Subtitle: Inhibitor of PI3K isoform p110α
Biological Activity: Biological Activity of PIK-75Description PIK-75 is an inhibitor of P13K with IC50 values of 5.8 nM, 76 nM, 0.51 μM and 1.3 μM for p110α, p110γ, p110δ and p110β, respectively. Targets p110α p110γ p110δ p110β DNA-PK IC50 5.8 nM 76 nM 0.
SMLES: CC1=C(C=C(C=C1)[N+](=O)[O-])S(=O)(=O)N(C)N=CC2=CN=C3N2C=C(C=C3)Br.Cl
CAS NO: 690270-29-2
Standard In CHIKey: Parasite inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C16H14BrN5O4S.HCl
M.Wt: 488.74
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/257/1/416
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Limited solubility
Storage:
Purity: >98%
Chemical Name: N-[(E)-(6-bromoimidazo[1,2-a]pyridin-3-yl)methylideneamino]-N,2-dimethyl-5-nitrobenzenesulfonamide;hydrochloride