Product Name: PIK-93
Subtitle: PI3Kγ/PI4KIIIβ/PI3Kα inhibitor
Biological Activity: Biological Activity of PIK-93Description PIK-93 is the first potent, synthetic inhibitor of PI3Kγ, PI4KIIIβ and PI3Kα with IC50 values of 16 nM, 19 nM and 39nM, respectively. Targets PI3Kγ PI4KIIIβ PI3Kα DNA-PK PI3Kδ IC50 16 nM 19 nM
SMLES: CC1=C(SC(=N1)NC(=O)C)C2=CC(=C(C=C2)Cl)S(=O)(=O)NCCO
CAS NO: 1268524-70-4
Standard In CHIKey: Mps1 inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C14H16ClN3O4S2
M.Wt: 389.88
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/257/2/668
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO > 10 mM
Storage:
Purity: >98%
Chemical Name: N-[5-[4-chloro-3-(2-hydroxyethylsulfamoyl)phenyl]-4-methyl-1,3-thiazol-2-yl]acetamide