Product Name: Varenicline tartrate
Subtitle: Subtype-selective agonist of α4β2 nicotinic receptors,orally active
Biological Activity: Biological Activity of Varenicline tartrate Orally active, subtype-selective partial agonist at α4β2 nicotinic receptors (Ki values are 0.06, 240, 322 and 3540 nM for α4β2, α3β4, α7, α1βγδ receptors r
SMLES: O[C@@H]([C@H](O)C(O)=O)C(O)=O.C1NCC2CC1c3cc4nccnc4cc23
CAS NO: 1311367-27-7
Standard In CHIKey: TWYFGYXQSYOKLK-WUUYCOTASA-NROS inhibitors
Standard InChI: InChI=1S/C13H13N3.C4H6O6/c1-2-16-13-5-11-9-3-8(6-14-7-9)10(11)4-12(13)15-1;5-1(3(7)8)2(6)4(9)10/h1-2,4-5,8-9,14H,3,6-7H2;1-2,5-6H,(H,7,8)(H,9,10)/t;1-,2-/m.0/s1
Typrof Compound: Alkaloids
Appearance: Powder
Formula: C13H13N3.C4H6O6
M.Wt: 361.35
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/256/3/1063
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in water and to 50 mM in DMSO
Storage: Desiccate at RT
Purity: ≥98%
Chemical Name: 7,8,9,10-Tetrahydro-6,10-methano-6H-pyrazino[2,3-h][3]benzazepine tartrate