Product Name: kb NB 142-70
Subtitle: Inhibitor of protein kinase D,selective
Biological Activity: Biological Activity of kb NB 142-70Selective protein kinase D (PKD) inhibitor (IC50 values are 28.3, 58.7 and 53.2 nM for PKD1, 2 and 3 respectively). More potent analog of CID 755673 with 7-fold greater inhibition. Inhibits prostrate cancer cell migratio
SMLES: C1CSC2=C(C(=O)N1)SC3=C2C=C(C=C3)O
CAS NO: 254750-02-2
Standard In CHIKey: PKD inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C11H9NO2S2
M.Wt: 251.32
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/251/1/105
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in DMSO
Storage: Store at RT
Purity: >98%
Chemical Name: 9-Hydroxy-3,4-dihydro-2H-[1]-benzothiolo[2,3-f][1,4]thiazepin-5-one