Product Name: ML161
Subtitle: PAR1 inhibitor
Biological Activity: Biological Activity of ML161Inhibitor of protease-activated receptor 1 (PAR1)-mediated platelet activation (IC50 = 0.26 μM for the inhibition of platelet P-selectin expression on human platelets). Thought to act allosterically. Also inhibits thrombin
SMLES: CCCC(=O)NC1=CC=CC(=C1)NC(=O)C2=CC=CC=C2Br
CAS NO: 1204669-58-8
Standard In CHIKey: Glucocorticoid Receptor inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C17H17BrN2O2
M.Wt: 361.23
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/251/2/586
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in DMSO and to 100 mM in ethanol
Storage: Store at +4℃
Purity: >98%
Chemical Name: 2-Bromo-N-[3-[(1-oxobutyl)amino]phenyl]benzamide