Product Name: Apatinib
Subtitle: VEGFR2 inhibitor, orally bioavailable, selective
Biological Activity: Biological Activity of ApatinibDescription Apatinib is an orally bioavailable, selective inhibitor of VEGFR2 with an IC50 value of 1 nM. Targets VEGFR2 RET c-Kit c-Src PDGFRα IC50 1 nM 13 nM 429 nM 530 nM >1 μM
SMLES:
CAS NO: 949912-58-7
Standard In CHIKey: CRAC Channel inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C25H27N5O4S
M.Wt: 493.58
General Tips: for obtaining a higher concentration: Please warm the tube at 37 ℃ for 10 minutes and/or shake it in the ultrasonic bath for a while. Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/275/1/368
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility:
Storage:
Purity: >98%
Chemical Name: